DG02852 | |
DG番号 | DG02852 |
分類 | DGroup |
名称 | CYP3A/CYP3A4 inhibitor TYPE Metabolism |
ステム | - |
構造式 | ![]() |
メンバー | DG01522 CYP3A4 inhibitor D00282 Clotrimazole (JP18/USP/INN) DG00017 Cimetidine D00295 Cimetidine (JP18/USP/INN) D03503 Cimetidine hydrochloride (USP) D10246 Omeprazole, clarithromycin and amoxicillin D08774 Amoxicillin hydrate, clarithromycin and lansoprazole D10519 Rabeprazole, amoxicillin and clarithromycin D10775 Vonoprazan, amoxicillin and clarithromycin DG00066 Aprepitant D02968 Aprepitant (JAN/USP/INN) D10895 Fosaprepitant (INN) D06597 Fosaprepitant dimeglumine (USAN); Fosaprepitant meglumine (JAN) D09394 Fidaxomicin (JAN/USAN) DG01283 Teneligliptin D08616 Teneligliptin (INN) D09756 Teneligliptin hydrobromide hydrate (JAN) D11968 Teneligliptin hydrobromide (JAN) DG03079 Berotralstat D11673 Berotralstat (USAN/INN) D11674 Berotralstat hydrochloride (JAN/USAN) DG00371 Fluconazole D00322 Fluconazole (JP18/USP/INN) D01429 Fosfluconazole (JAN/INN) D01980 Luliconazole (JAN/USAN/INN) DG00452 Bromocriptine D03165 Bromocriptine (USAN/INN) D00780 Bromocriptine mesylate (USP); Bromocriptine mesilate (JP18) DG00461 Ethinylestradiol D00554 Ethinyl estradiol (USP); Ethinylestradiol (JP18/INN) D07928 Ethinylestradiol propanesulfonate DG01903 Midecamycin D01339 Midecamycin (JP18/INN) D01636 Midecamycin acetate (JP18) DG00604 Josamycin D01235 Josamycin (JP18/USAN/INN) D05351 Josamycin propionate (JP18) D01322 Troleandomycin (USAN/INN); Triacetyloleandomycin (JAN) DG00605 Clarithromycin D00276 Clarithromycin (JP18/USP/INN) D07710 Clarithromycin lactobionate D00854 Quinupristin and dalfopristin D00350 Itraconazole (JP18/USP) D02555 Posaconazole (JAN/USAN/INN) DG00654 Indinavir C07051 Indinavir D03833 Indinavir (USAN) D00897 Indinavir sulfate (USP) D02861 Indinavir sulfate ethanolate (JAN) DG00655 Nelfinavir D08259 Nelfinavir (INN) D00899 Nelfinavir mesylate (USAN/INN); Nelfinavir mesilate (JAN) DG00656 Fosamprenavir D02497 Fosamprenavir (INN) D02867 Fosamprenavir calcium hydrate (JAN) D03835 Fosamprenavir calcium (USAN) D03837 Fosamprenavir sodium (USAN) DG00657 Atazanavir D07471 Atazanavir (INN) D01276 Atazanavir sulfate (JAN/USAN) DG00659 Darunavir D03656 Darunavir (USAN/INN) D06478 Darunavir ethanolate (JAN) D12637 Darunavir hydrate D09012 Telaprevir (JAN/USAN/INN) D10582 Dasabuvir, ombitasvir, paritaprevir and ritonavir D10745 Ombitasvir, paritaprevir and ritonavir D00753 Sirolimus (JAN/USAN/INN) D00961 Bicalutamide (JP18/USP/INN) D00960 Anastrozole (JP18/USP/INN) D00184 Cyclosporine (USP); Ciclosporin (JP18) D05928 Stiripentol (JAN/USAN/INN) D04641 Istradefylline (JAN/USAN/INN) DG00946 Fluvoxamine D07984 Fluvoxamine (INN) D00824 Fluvoxamine maleate (JP18/USP) D08837 Aclidinium bromide (JAN/USAN/INN) D00707 Fomepizole (JAN/USAN/INN) D09799 Carotegrast methyl (JAN) DG00004 Miconazole D00416 Miconazole (JP18/USP/INN) D00882 Miconazole nitrate (JP18/USP) DG00018 Ranitidine D00422 Ranitidine (USAN/INN) D00673 Ranitidine hydrochloride (JP18/USP) D05699 Ranitidine bismuth citrate (USAN) D09017 Ticagrelor (JAN/USAN/INN) DG01419 Fostamatinib D09347 Fostamatinib (USAN) D09348 Fostamatinib disodium (USAN); Fostamatinib sodium hydrate (JAN) DG00207 Dronedarone D02537 Dronedarone (INN) D03914 Dronedarone hydrochloride (USP) DG00276 Conivaptan D07748 Conivaptan (INN) D01236 Conivaptan hydrochloride (JAN/USAN) DG00328 Mibefradil D08217 Mibefradil (INN) D05024 Mibefradil dihydrochloride (USAN) DG02844 Ravuconazole D02556 Ravuconazole (prop.INN) D10762 Fosravuconazole L-lysine ethanolate (JAN) DG00436 Erythromycin D00140 Erythromycin (JP18/USP/INN) D00851 Erythromycin estolate (USP); Erythromycin estorate (JAN) D01361 Erythromycin ethylsuccinate (JP18/USP) D02009 Erythromycin lactobionate (JP18/USP) D02184 Erythromycin stearate (JP18/USP) D02523 Erythromycin acistrate (USAN) D02524 Erythromycin gluceptate (USP) D02525 Erythromycin propionate (USAN) D03098 Berythromycin (USAN/INN) D04054 Erythromycin salnacedin (USAN) D07909 Erythromycin thiocyanate D07910 Erythromycin stinoprate (INN) D00585 Mifepristone (JAN/USAN/INN) D12586 Mifepristone and misoprostol D01078 Telithromycin (JAN/USAN/INN) DG00620 Norfloxacin D00210 Norfloxacin (JP18/USP/INN) D08287 Norfloxacin nicotinate D00578 Voriconazole (JP18/USP/INN) D00427 Ritonavir (JAN/USP/INN) D00894 Amprenavir (JAN/USAN/INN) D12269 Nirmatrelvir and ritonavir DG00662 Delavirdine D07782 Delavirdine (INN) D00895 Delavirdine mesylate (USAN); Delavirdine mesilate (JAN) D08876 Boceprevir (INN/USAN) DG01246 Simeprevir D10081 Simeprevir (JAN/USAN) D10469 Simeprevir sodium (JAN) DG01669 Daclatasvir D10065 Daclatasvir (USAN) D10105 Daclatasvir dihydrochloride (USAN); Daclatasvir hydrochloride (JAN) DG03051 Grazoprevir D11565 Grazoprevir (USAN/INN) D10639 Grazoprevir (USAN); Grazoprevir hydrate (JAN) D10756 Elvitegravir, cobicistat, emtricitabine and tenofovir disoproxil D02498 Lopinavir and ritonavir D10753 Atazanavir and cobicistat D10801 Letermovir (JAN/USAN/INN) D09731 Crizotinib (JAN/USAN/INN) D10926 Entrectinib (JAN/USAN/INN) DG00942 Fluoxetine D00326 Fluoxetine (USAN/INN) D00823 Fluoxetine hydrochloride (JAN/USP) D09881 Cobicistat (JAN/USAN/INN) D11920 Pimitespib (JAN) D11970 Ritlecitinib tosylate (USAN); Ritlecitinib tosilate (JAN) DG01840 Isavuconazonium D10644 Isavuconazonium (USAN) D10643 Isavuconazonium sulfate (JAN/USAN) DG03269 Ensitrelvir D12619 Ensitrelvir (USAN/INN) D12353 Ensitrelvir fumarate (USAN); Ensitrelvir fumaric acid (JAN) D01425 Lopinavir (JAN/USP/INN) D05152 Netupitant (USAN/INN) |
上位グループ | Metabolizing enzyme inhibitor |
注釈1 | - |
注釈2 | - |