DG02924 | |
DG番号 | DG02924 |
分類 | DGroup |
名称 | UGT substrate TYPE Metabolism |
ステム | - |
構造式 | ![]() |
メンバー | DG03183 UGT1A1 substrate D11051 Vericiguat (JAN/USAN/INN) DG00666 Raltegravir D06676 Raltegravir (INN) D07133 Raltegravir potassium (JAN/USAN) DG00667 Dolutegravir D10066 Dolutegravir (USAN) D10113 Dolutegravir sodium (JAN/USAN) DG01628 Cabotegravir D10548 Cabotegravir (JAN/USAN/INN) D10549 Cabotegravir sodium (JAN/USAN) D10600 Dolutegravir, abacavir and lamivudine D11282 Dolutegravir sodium and rilpivirine hydrochloride DG03049 Tecovirimat D09390 Tecovirimat (USAN/INN) D11557 Tecovirimat monohydrate DG03165 Lenacapavir D12161 Lenacapavir (USAN/INN) D12162 Lenacapavir sodium (JAN/USAN) DG00726 Irinotecan D08086 Irinotecan (INN) D01061 Irinotecan hydrochloride (USP); Irinotecan hydrochloride hydrate (JP18) D10642 Irinotecan sucrosofate (USAN) DG01414 Selumetinib D09666 Selumetinib (USAN/INN) D10024 Selumetinib sulfate (JAN/USAN) D08870 Belinostat (USAN/INN) DG01058 Olodaterol D10145 Olodaterol (USAN/INN) D10020 Olodaterol hydrochloride (JAN/USAN) D03669 Deferasirox (JAN/USAN/INN) D11966 Cabotegravir and rilpivirine DG03184 UGT1A3 substrate D10459 Empagliflozin (JAN/USAN/INN) D09994 Selexipag (JAN/USAN/INN) DG01414 Selumetinib D09666 Selumetinib (USAN/INN) D10024 Selumetinib sulfate (JAN/USAN) D03669 Deferasirox (JAN/USAN/INN) DG03182 UGT1A4 substrate D06273 Imidafenacin (JAN/INN) DG03049 Tecovirimat D09390 Tecovirimat (USAN/INN) D11557 Tecovirimat monohydrate D10560 Idelalisib (JAN/USAN/INN) DG02960 Pexidartinib D11270 Pexidartinib (USAN/INN) D11271 Pexidartinib hydrochloride (JAN/USAN) D00354 Lamotrigine (JAN/USP/INN) DG03185 UGT1A7 substrate D10915 Cannabidiol (USAN/INN) DG01058 Olodaterol D10145 Olodaterol (USAN/INN) D10020 Olodaterol hydrochloride (JAN/USAN) DG03186 UGT1A8 substrate D10459 Empagliflozin (JAN/USAN/INN) DG03188 UGT1A9 substrate D11066 Ertugliflozin and sitagliptin DG00122 Dapagliflozin D08897 Dapagliflozin (USAN/INN) D09763 Dapagliflozin propanediol (USAN); Dapagliflozin propylene glycolate hydrate (JAN) D09592 Canagliflozin (USAN/INN); Canagliflozin hydrate (JAN) D10459 Empagliflozin (JAN/USAN/INN) DG02836 Ertugliflozin D10313 Ertugliflozin (USAN/INN) D11043 Ertugliflozin pidolate D10669 Sotagliflozin (USAN/INN) D10593 Roxadustat (JAN/USAN/INN) D11051 Vericiguat (JAN/USAN/INN) DG01628 Cabotegravir D10548 Cabotegravir (JAN/USAN/INN) D10549 Cabotegravir sodium (JAN/USAN) DG00720 Regorafenib D10138 Regorafenib (USAN/INN) D10137 Regorafenib hydrate (JAN) D11817 Deucravacitinib (JAN/USAN) D10915 Cannabidiol (USAN/INN) D05768 Rotigotine (JAN/USAN/INN) DG00956 Viloxazine D08673 Viloxazine (INN) D02572 Viloxazine hydrochloride (USAN) DG01058 Olodaterol D10145 Olodaterol (USAN/INN) D10020 Olodaterol hydrochloride (JAN/USAN) D10865 Bexagliflozin (USAN) D10897 Teneligliptin and canagliflozin D11966 Cabotegravir and rilpivirine DG03189 UGT2B4 substrate D09592 Canagliflozin (USAN/INN); Canagliflozin hydrate (JAN) DG00814 Dihydrocodeine D07831 Dihydrocodeine (INN) D01481 Dihydrocodeine phosphate (JP18) D03825 Dihydrocodeine bitartrate (USP) D07832 Dihydrocodeine thiocyanate D08695 dl-Methylephedrine hydrochloride, dihydrocodeine phosphate, diprophylline, diphenhydramine salicylate, acetaminophen and bromovalerylurea D11150 Cenobamate (USAN/INN) DG01076 Codeine C06174 Codeine D00195 Codeine (USP) D02101 Codeine phosphate (USP); Codeine phosphate hydrate (JP18) D03579 Codeine polistirex (USAN) D03580 Codeine sulfate (USP) D07740 Codeine hydrochloride D12312 Codeine phosphate and chlorpheniramine maleate D12313 Chlorpheniramine polistirex and codeine polistirex D04313 Dihydrocodeine phosphate, dl-methylephedrine hydrochloride and Chlorpheniramine maleate D04338 Dihydrocodeine phosphate, ephedrine hydrochloride and ammmonium chloride D08697 Platycodon fluidextract, glycyrrhiza extract, plantago herb extract, peony root extract and dihydrocodeine phosphate D10897 Teneligliptin and canagliflozin D11851 Butalbital, acetaminophen, caffeine and codeine phosphate D11860 Butalbital, aspirin, caffeine and codeine DG03190 UGT2B7 substrate D11066 Ertugliflozin and sitagliptin D10459 Empagliflozin (JAN/USAN/INN) DG02836 Ertugliflozin D10313 Ertugliflozin (USAN/INN) D11043 Ertugliflozin pidolate DG01248 Ipragliflozin D10196 Ipragliflozin (INN) D10200 Ipragliflozin L-proline (JAN) D09994 Selexipag (JAN/USAN/INN) DG03004 Asciminib D11403 Asciminib (USAN/INN) D11404 Asciminib hydrochloride (JAN/USAN) DG00814 Dihydrocodeine D07831 Dihydrocodeine (INN) D01481 Dihydrocodeine phosphate (JP18) D03825 Dihydrocodeine bitartrate (USP) D07832 Dihydrocodeine thiocyanate D08695 dl-Methylephedrine hydrochloride, dihydrocodeine phosphate, diprophylline, diphenhydramine salicylate, acetaminophen and bromovalerylurea D10915 Cannabidiol (USAN/INN) D11150 Cenobamate (USAN/INN) D00365 Lorazepam (JP18/USP/INN) DG01058 Olodaterol D10145 Olodaterol (USAN/INN) D10020 Olodaterol hydrochloride (JAN/USAN) DG01076 Codeine C06174 Codeine D00195 Codeine (USP) D02101 Codeine phosphate (USP); Codeine phosphate hydrate (JP18) D03579 Codeine polistirex (USAN) D03580 Codeine sulfate (USP) D07740 Codeine hydrochloride D12312 Codeine phosphate and chlorpheniramine maleate D12313 Chlorpheniramine polistirex and codeine polistirex D04313 Dihydrocodeine phosphate, dl-methylephedrine hydrochloride and Chlorpheniramine maleate D04338 Dihydrocodeine phosphate, ephedrine hydrochloride and ammmonium chloride D08697 Platycodon fluidextract, glycyrrhiza extract, plantago herb extract, peony root extract and dihydrocodeine phosphate D11064 Sitagliptin and ipragliflozin D11851 Butalbital, acetaminophen, caffeine and codeine phosphate D11860 Butalbital, aspirin, caffeine and codeine DG03187 UGT2B15 substrate D05768 Rotigotine (JAN/USAN/INN) D00365 Lorazepam (JP18/USP/INN) DG00956 Viloxazine D08673 Viloxazine (INN) D02572 Viloxazine hydrochloride (USAN) DG03181 UGT2B17 substrate DG03004 Asciminib D11403 Asciminib (USAN/INN) D11404 Asciminib hydrochloride (JAN/USAN) D11954 Belzutifan (JAN/USAN/INN) DG00081 Tegaserod D06056 Tegaserod (USAN/INN) D02730 Tegaserod maleate (USAN) D01854 Mitiglinide calcium hydrate (JP18) DG00229 Milrinone D00417 Milrinone (JAN/USP/INN) D02085 Milrinone lactate DG00339 Benazepril D07499 Benazepril (INN) D00620 Benazepril hydrochloride (JAN/USP) D00627 Telmisartan (JP18/USP/INN) D10480 Irbesartan and trichlormethiazide D09219 Telmisartan and hydrochlorothiazide (JP18) D10805 Telmisartan, amlodipine and hydrochlorothiazide D09743 Telmisartan and amlodipine besilate (JP18) DG01548 Fenofibrate D00565 Fenofibrate (JP18/USP/INN) D08890 Choline fenofibrate (USAN/INN) D01966 Ezetimibe (JAN/USP/INN) D01965 Silodosin (JP18/INN) D12137 Elagolix, estradiol and norethisterone DG02839 Osilodrostat D11061 Osilodrostat (USAN/INN) D11062 Osilodrostat phosphate (JAN/USAN) D11521 Lamivudine, nevirapine and zidovudine DG00714 Dasatinib D03658 Dasatinib (JAN/INN) D06414 Dasatinib (USAN); Dasatinib hydrate (JAN) D12609 Dasatinib laurylsulfate (USAN) DG01374 Nintedanib D10481 Nintedanib (USAN/INN) D10396 Nintedanib esylate (USAN); Nintedanib ethanesulfonate (JAN) D06320 Vorinostat (JAN/USAN) D11222 Selinexor (USAN/INN) DG01829 Esketamine D07283 Esketamine (USAN/INN) D10627 Esketamine hydrochloride (JAN/USAN) DG00810 Morphine D08233 Morphine (BAN) D00842 Morphine sulfate (USP); Morphine sulfate hydrate (JP18) D02271 Morphine hydrochloride hydrate (JP18) D08234 Morphine tartrate DG00811 Hydromorphone D08047 Hydromorphone (INN) D00839 Hydromorphone hydrochloride (JAN/USP) DG00826 Tapentadol D06007 Tapentadol (USAN/INN) D10199 Tapentadol hydrochloride (JAN) DG00963 Desvenlafaxine D07793 Desvenlafaxine (INN) D02570 Desvenlafaxine succinate (USAN); Desvenlafaxine succinate hydrate (JAN) D11619 Desvenlafaxine succinate anhydrous DG01052 Formoterol D07990 Formoterol (INN) D01373 Formoterol fumarate (USP) D05277 Formoterol fumarate hydrate (JP18) D09595 Budesonide and formoterol fumarate dihydrate D10506 Fluticasone propionate and formoterol fumarate hydrate D11857 Aclidinium bromide and formoterol fumarate D10744 Tiotropium and olodaterol D11520 Ezetimibe and rosuvastatin |
上位グループ | Metabolizing enzyme substrate |
注釈1 | - |
注釈2 | - |